• Patent

Cocaine receptor binding ligands


Carroll, F. (1998). IPC No. U.S.Cocaine receptor binding ligands (Patent No. 5736123.)

Novel compounds useful as intermediates in the synthesis ofcompounds having high affinity for specific cocaine receptors inthe brain have the formula ##STR1## wherein R is (CH.sub.2).sub.nCH.sub.2 Y, and wherein Y is H or F, X is a pharmaceuticallyacceptable anion, and wherein Sn (R.sup.1, R.sup.2, R.sup.3) isortho, meta or para and wherein R.sup.1, R.sup.2, R.sup.3 areindependently alkyl of 1-6 carbon atoms and n is an integer of0-5.