Pyrazole Derivatives as Cannabinoid Receptor 1 Antagonists
Fulp, A., Maitra, R., Zhang, Y., & Seltzman, H. (2015). Pyrazole Derivatives as Cannabinoid Receptor 1 Antagonists. (U.S. Patent No. 9133128). http://patft.uspto.gov/netacgi/nph-Parser?patentnumber=9133128
Abstract
The invention provides compounds capable of acting as antagonists at cannabanoid receptors according to the following formula; Such compounds may be used to treat conditions for which the cannabinoid receptor system has been implicated, such as obesity, liver disease, diabetes, pain, and inflammation.
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