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Search Results

Showing results 21 to 40 of 53.

Article

Reversal of Ethanol-induced Intoxication by a Novel Modulator of Gβγ Protein Potentiation of the Glycine Receptor

September 02, 2016
Article

Clozapine metabolites protect dopaminergic neurons through inhibition of microglial NADPH oxidase

May 16, 2016
Article

FL118, a novel camptothecin derivative, is insensitive to ABCG2 expression and shows improved efficacy in comparison with irinotecan in colon and lung cancer models with ABCG2–induced resistance

April 01, 2015
Article

Synthesis, Pharmacological Characterization, and Structure-Activity Relationship Studies of Small Molecular Agonists for the Orphan GPR88 Receptor

July 01, 2014
Article

Discovery of N-{4-[(3-Hydroxyphenyl)-3-methylpiperazin-1-yl]methyl-2-methylpropyl}-4-phenoxybenzamide Analogues as Selective Kappa Opioid Receptor Antagonists

June 13, 2013
Article

The GPR88 receptor agonist 2-PCCA does not alter the behavioral effects of methamphetamine in rats

January 01, 2013
Article

Synthesis and antihormonal properties of novel 11ß-benzoxazole-substituted steroids

February 01, 2012
Article

Synthesis and structure-activity relationship of 3beta-(4-alkylthio, -methylsulfinyl, and -methylsulfonylphenyl)tropane and 3beta-(4-alkylthiophenyl)nortropane derivatives for monoamine transporters

July 15, 2009
Article

Synthesis and structure-activity relationship of 3ß-(4-alkylthio, -methylsulfinyl, and -methylsulfonylphenyl)tropane and 3ß-(4-alkylthiophenyl)nortropane derivatives for monoamine transporters

July 01, 2009
Article

A short and efficient synthesis of 3-{2-[2-(bromomethyl)thiazol-4-yl]ethynyl}-5-fluorobenzonitrile:: A precursor for PET radioligand [F-18]SP203

June 01, 2009
Article

Synthesis of carnosine-d7 and anserine-d4 for use as internal standards in liquid chromatography-mass spectrometry

January 01, 2009
Article

Development of 3-phenyltropane analogues with high affinity for the dopamine and serotonin transporters and low affinity for the norepinephrine transporter

December 25, 2008
Article

Development of 3-phenyltropane analogs with high affinity for the dopamine and serotonin transporters and low affinity for the norepinephrine transporter

December 01, 2008
Article

Synthesis and monoamine transporter binding properties of 2beta-[3'-(substituted benzyl)isoxazol-5-yl]- and 2beta-[3'-methyl-4'-(substituted phenyl)isoxazol-5-yl]-3beta-(substituted phenyl)tropanes

July 15, 2008
Article

Synthesis and monoamine transporter binding properties of 2ß-[3'-(substituted benzyl)isoxazol-5-yl]- and 2ß-[3'-methyl-4'-(substituted phenyl)isoxazol-5-yl]-3ß-(substituted phenyl)tropanes

July 01, 2008
Article

Synthesis and receptor binding properties of 2beta-alkynyl and 2beta-(1,2,3-triazol)substituted 3beta-(substituted phenyl)tropane derivatives

May 15, 2008
Article

Synthesis and receptor binding properties of 2ß-alkynyl and 2ß-(1,2,3-triazol)­substituted 3ß-(substituted phenyl)tropane derivatives

May 01, 2008
Article

Convenient synthesis of tolcapone, a selective catechol-O-methyltransferase inhibitor

January 01, 2008
Article

Practical synthesis of p-aminophenethylspiperone (NAPS), a high-affinity, selective D-2-dopamine receptor antagonist

January 01, 2008
Article

Synthesis and identification of novel 11beta-aryl-4',5'-dihydrospiro[estra-4,9-diene-17beta,4'-oxazole] analogs with dissociated antiprogesterone activities

November 01, 2007