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Search Results

Showing results 1 to 20 of 62.

Article

Diarylureas as Allosteric Modulators of the Cannabinoid CB1 Receptor: Structure-Activity Relationship Studies on 1-(4-Chlorophenyl)-3-{3-[6-(pyrrolidin-1-yl)pyridin-2-yl]phenyl}urea (PSNCBAM-1)

September 25, 2014
Article

Fragmentations of (E)- and (Z)-isomers of 2-methylbuten-1-yl(aryl) iodonium triflates: Competing mechanisms for enol triflate formation

July 25, 2003
Patent

Phenylmorpholines and Analogues Thereof

April 11, 2017
Article

Development of norepinephrine transporter reuptake inhibition assays using SK-N-BE(2)C cells

May 01, 2018
Article

Synthesis and pharmacological validation of a novel radioligand for the orphan GPR88 receptor

January 15, 2023
Patent

Vinylogous phenethylamines as neurotransmitter releasers

January 26, 2021
Article

Identification of 2-({[1-(4-Fluorophenyl)-5-(2-methoxyphenyl)-1H-pyrazol-3-yl]carbonyl)}amino)tricyclo[3.3.1.13,7]decane-2-carboxylic Acid (NTRC-844) as a selective antagonist for the rat neurotensin receptor type 2

September 21, 2016
Article

Novel diarylurea based allosteric modulators of the cannabinoid CB1 receptor: Evaluation of importance of 6-pyrrolidinylpyridinyl substitution

September 14, 2017
Chapter

Interrogating the Activity of Ligands at Monoamine Transporters in Rat Brain Synaptosomes

August 01, 2016
Article

Synthesis of a bistetrahydrofuran C17-C32 fragment of the polyether antibiotic ionomycin

September 14, 2006
Article

Discovery of a potent, selective, and brain-penetrant small molecule that activates the orphan receptor GPR88 and reduces alcohol intake

August 09, 2018
Article

In vitro and in vivo evaluation of pellotine: A hypnotic lophophora alkaloid

October 13, 2023
Article

Design, synthesis and pharmacological evaluation of 4-hydroxyphenylglycine and 4-hydroxyphenylglycinol derivatives as GPR88 agonists

January 15, 2017
Article

Discovery of novel proline-based neuropeptide FF receptor antagonists

October 18, 2017
Article

Potent and selective tetrahydroisoquinoline kappa opioid receptor antagonists of lead compound (3 R)- N-[1 R)-1-(Cyclohexylmethyl)-2-methylpropyl]-7-hydroxy-1,2,3,4-tetrahydroisoquinoline-3-carboxamide (CDTic)

September 13, 2018
Article

Discovery of a novel small molecule agonist scaffold for the APJ receptor

August 15, 2016
Article

Validation of a high-throughput calcium mobilization assay for the human trace amine-associated receptor 1

January 01, 2021
Article

Truncated orexin peptides: structure–activity relationship studies

December 01, 2013
Article

Evaluation of amide bioisosteres leading to 1,2,3-triazole containing compounds as GPR88 agonists: Design, synthesis, and structure-activity relationship studies

August 26, 2021
Article

Fluorinated phenmetrazine "legal highs" act as substrates for high-affinity monoamine transporters of the SLC6 family

May 15, 2018