• Journal Article

Rapid in-plate generation of benzimidazole libraries and amide formation using EEDQ

Citation

Thomas, J., Fall, M., Cooper, J., Burgess, J., & Carroll, F. (1997). Rapid in-plate generation of benzimidazole libraries and amide formation using EEDQ. Tetrahedron Letters, 38(29), 5099-5102.

Abstract

A solution phase method for the preparation of etonitazene-related benzimidazoles and a general method for the preparation of amide derivatives in 96-well format have been developed for the generation of libraries of compounds in parallel. (C) 1997 Elsevier Science Ltd